Issue Date | Title | Author(s) | Relation | scopus | WOS | Fulltext/Archive link |
2010 | Combination of bifunctional alkylating agent and arsenic trioxide synergistically suppresses the growth of drug-resistant tumor cells. | Lee, PC; Kakadiya, R; Su, TL; Lee, TC | NEOPLASIA 12(5), 376-87 | | | |
2011 | Design, synthesis and antitumor evaluation of phenyl N-mustard-quinazoline conjugates. | Marvania, B; Lee, PC; Chaniyara, R; Dong, H; Suman, S; Kakadiya, R; Chou, TC; Lee, TC; Shah, A; Su, TL | Bioorganic & medicinal chemistry 19(6), 1987-1998 | | | |
2011 | Design, synthesis, and biological evaluation of novel water-soluble N-mustards as potential anticancer agents. | Kapuriya, N; Kakadiya, R; Dong, H; Kumar, A; Lee, PC; Zhang, X; Chou, TC; Lee, TC; Chen, CH; Lam, K; Marvania, B; Shah, A; Su, TL | BIOORGANIC & MEDICINAL CHEMISTRY 19(1), 471-485 | | | |
2013 | Determination of tissue distribution of potent antitumor agent ureidomustin (BO-1055) by HPLC and its pharmacokinetic application in rats. | Chien, SI; Yen, JC; Kakadiya, R; Chen, CH; Lee, TC; Su, TL; Tsai, TH | Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 917-918, 62-70 | | | |
2012 | Multidrug-resistant cells overexpressing P-glycoprotein are susceptible to DNA crosslinking agents due to attenuated Src/nuclear EGFR cascade-activated DNA repair activity | Lee, PC; Lee, HJ; Kakadiya, R; Sanjiv, K; Su, TL; Lee, TC | Oncogene | | | |
2011 | Novel 2-substituted quinolin-4-yl-benzenesulfonate derivatives: synthesis, antiproliferative activity, and inhibition of cellular tubulin polymerization. | Kakadiya, R; Wu, YC; Dong, H; Kuo, HH; Yih, LH; Chou, TC; Su, TL | ChemMedChem 6(6), 1119-1129 | | | |
- | Novel Antitumor Indolizino[6,7-b]indoles with Multiple Modes of Action: DNA Cross-Linking and Topoisomerase I and II Inhibition. | Chaniyara, R; Tala, S; Chen, CW; Zang, X; Kakadiya, R; Lin, LF; Chen, CH; Chien, SI; Chou, TC; Tsai, TH; Lee, TC; Shah, A; Su, TL. | JOURNAL OF MEDICINAL CHEMISTRY | | | |
2011 | Novel bifunctional alkylating agents, 5,10-dihydropyrrolo[1,2-b]isoquinoline derivatives, synthesis and biological activity. | Chaniyara, R; Kapuriya, N; Dong, H; Lee, PC; Suman, S; Marvania, B; Chou, TC; Lee, TC; Kakadiya, R; Shah, A; Su, TL | Bioorganic & medicinal chemistry 19(1), 275-286 | | | |
2014 | PI3K Inhibition Augments the Therapeutic Efficacy of a 3a-aza-Cyclopenta[alpha]indene Derivative in Lung Cancer Cells. | Sanjiv, K; Chen, CW; Kakadiya, R; Tala, S; Suman, S; Wu, MH; Chen, YH; Su, TL; Lee, TC | Translational oncology 7(2), 256-266.e5 | | | |
2009 | Potent antitumor bifunctional DNA alkylating agents, synthesis and biological activities of 3a-aza-cyclopenta[a]indenes. | Kakadiya, R; Dong, H; Lee, PC; Kapuriya, N; Zhang, X; Chou, TC; Lee, TC; Kapuriya, K; Shah, A; Su, TL | Bioorganic & medicinal chemistry 17(15), 5614-26 | | | |
2008 | Potent bifunctional DNA alkylating agents, derivatives of 3a-aza-cyclopenta[a]indenes against human solid tumor xenografts. | Su, T. -L; Kakadiya, R; Kapuriya, N; Zhang, X; Chou, T. -C. | | | | |
2010 | Potent DNA-directed alkylating agents. Synthesis and biological activity of phenyl N-mustard-quinoline conjugates having a urea or hydrazinecarboxamide linker | Kakadiya, R; Dong, H; Kumar, A; Narsinh, D; Zhang, X; Chou, TC; Lee, TC; Shah, A; Su, TL | BIOORGANIC & MEDICINAL CHEMISTRY 18(6), 2285-2299 | | | |
2010 | Potent DNA-directed alkylating agents: Synthesis and biological activity of phenyl N-mustard-quinoline conjugates having a urea or hydrazinecarboxamide linker. | Kakadiya, R; Dong, H; Kumar, A; Narsinh, D; Zhang, X; Chou, TC; Lee, TC; Shah, A; Su, TL | Bioorganic & medicinal chemistry 18(6), 2285-99 | | | |
2015 | Repairing of N-mustard derivative BO-1055 induced DNA damage requires NER, HR, and MGMT-dependent DNA repair mechanisms. | Kuo, CY; Chou, WC; Wu, CC; Wong, TS; Kakadiya, R; Lee, TC; Su, TL; Wang, HC | Oncotarget 6(28), 25770-83 | | | |
2012 | Synthesis and antitumor evaluation of novel Benzo[d]pyrrolo[2,1-b]thiazole derivatives | Chaniyara, R; Tala, S; Chen, CW; Lee, PC; Kakadiya, R; Dong, H; Marvania, B; Chen, CH; Chou, TC; Lee, TC; Shah, A; Su, TL | Eur. J. Med. Chem. 53, 28-40 | | | |
2012 | Synthesis and antitumor evaluation of novel benzo[d]pyrrolo[2,1-b]thiazole derivatives. | Chaniyara, R; Tala, S; Chen, CW; Lee, PC; Kakadiya, R; Dong, H; Marvania, B; Chen, CH; Chou, TC; Lee, TC; Shah, A; Su, TL | European journal of medicinal chemistry 53, 28-40 | | | |
2008 | Synthesis and biological activity of stable and potent antitumor agents, aniline nitrogen mustards linked to 9-anilinoacridines via a urea linkage. | Kapuriya, N; Kapuriya, K; Zhang, X; Chou, TC; Kakadiya, R; Wu, YT; Tsai, TH; Chen, YT; Lee, TC; Shah, A; Naliapara, Y; Su, TL | Bioorganic & medicinal chemistry 16(10), 5413-23 | | | |
2009 | Synthesis and in vitro cytotoxicity of 9-anilinoacridines bearing N-mustard residue on both anilino and acridine rings. | Chen, CH; Lin, YW; Zhang, X; Chou, TC; Tsai, TJ; Kapuriya, N; Kakadiya, R; Su, TL | European journal of medicinal chemistry 44(7), 3056-9 | | | |
2011 | Synthesis of new tetracyclic 7-oxo-pyrido[3,2,1-de]acridine derivatives | Chen, CH; Lin, YW; Kakadiya, R; Kumar, A; Chen, YT; Lee, TC; Su, TL | Tetrahedron 67(33), 5883-5893 | | | |
2012 | The novel DNA alkylating agent BO-1090 suppresses the growth of human oral cavity cancer in xenografted and orthotopic mouse models. | Sanjiv, K; Su, TL; Suman, S; Kakadiya, R; Lai, TC; Wang, HY; Hsiao, M; Lee, TC | International Journal of Cancer 130(6), 1440-1450 | | | |